Dipiaron is an oral agonist of the GPR119 receptor, which is a new validated target for T2DM therapy. Due to low systemic availability, it stimulates GPR119 in specialized L- and K-cells of the epithelium of the gastrointestinal tract.
It belongs to the group of modern drugs, such as GLP-1 analogues and DPP-4 inhibitors, which stimulate the production of incretins. The drugs of this group cause pleiotropic effects in the body: a decrease in the risk of cardiovascular complications of diabetes, endothelial, neuro- and cardioprotective effects
Dipiaron is an innovative highly effective non-injectable drug for the treatment of type 2 diabetes mellitus (T2DM), which helps to reduce the incidence of systemic side effects and complications of the disease.